血管生成库

Angiogenesis related Compound Library
产品编号: L4800

血管生成是正常生长和发育过程以及伤口愈合和肉芽组织形成过程中的基本事件,然而异常的血管生成将导致各种疾病,例如肿瘤、糖尿病、免疫病、先兆子痫、肢体缺血等。因此,血管生成已成为治疗这些疾病的药物靶点。例如,血管生成与癌症发生密切相关,肿瘤通过分泌各种生长因子(例如VEGF)和蛋白质诱导毛细血管生成进入肿瘤,为癌细胞提供氧气和其他必需的营养物质,并及时运走代谢废物,血管生成也是肿瘤扩散或转移所必需的。因此血管生成抑制剂用于治疗癌症。此外,诱导血管生成,建立新的侧支循环是治疗缺血性心脑血管疾病(冠心病、脑卒中等)的极佳治疗方式。有效新生血管靶分子的筛选为相关疾病研究带来了广阔前景。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L4800
产品编号: L4800
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品描述:
  • 2300个高潜力的抑制或促进血管生成的小分子集合,可用于药物靶点开发、血管生成机理研究的高通量筛选,高内涵筛选;
  • 包含了目前研究较多潜力的血管生成通路以及S1P、VEGFR、PDGF等相关靶点的热门产品;
  • 包含了Sunitinib Malate、Lenalidomide、sorafenib、Erlotinib等研究成熟的上市药物,以及Vatalanib、Orantinib、2-Methoxyestradiol(Panzem)、Celecoxib等临床药物;
  • 是研究血管生成机理以及药物靶向研究的有效工具;
  • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。
化合物库定制
我们的化合物库可以灵活定制! 了解更多
化合物库咨询
验证码
化合物库组成
5-HT Receptor
Apoptosis
Autophagy
PI3K
EGFR
VEGFR
COX
TNF
JAK
mTOR
Akt
p38 MAPK
FLT
Src
Dopamine Receptor
PDGFR
AMPK
FGFR
GSK-3
Bcr-Abl
ALK
c-Kit
TGF-beta/Smad
CDK
Adrenergic Receptor
HIF/HIF Prolyl-Hydroxylase
NF-κB
MMP
Antibacterial
Endogenous Metabolite
HIF
Histamine Receptor
IL Receptor
Tyrosine Kinases
CXCR
ERK
Potassium Channel
DNA-PK
FAK
c-Met/HGFR
AChR
S6 Kinase
HER
STAT
ATM/ATR
Syk
Parasite
Aurora Kinase
Raf
c-RET
Reactive Oxygen Species
Serotonin Transporter
PDK
IGF-1R
Norepinephrine
PKC
JNK
Gamma-secretase
HIV Protease
BTK
Antibiotic
PKA
Caspase
Influenza Virus
Interleukin
Mitophagy
PPAR
MEK
TAM Receptor
c-Fms
MAPK
NO Synthase
Calcium Channel
Casein Kinase
PI4K
Antifungal
DNA/RNA Synthesis
Antioxidant
Beta Amyloid
Cytochromes P450
Drug Metabolite
Lipoxygenase
NOS
Sodium Channel
Trk receptor
Ferroptosis
Microtubule Associated
PDE
Virus Protease
Wnt/beta-catenin
Chk
Dehydrogenase
HDAC
IκB/IKK
ROS
Bcl-2 Family
PARP
ROS Kinase
CSF-1R
GABA Receptor
Phosphatase
Prostaglandin Receptor
ROCK
Tyrosinase
Cholinesterase (ChE)
Ephrin Receptor
Nrf2
PYK2
SIK
Antiviral
CCR
DYRK
HCV Protease
MAO
MELK
MLK
Opioid Receptor
P-gp
PTEN
Serine/threonin kinase
Sigma receptor
TLR
Adenosine Receptor
Antifection
Carbonic Anhydrase
Histone Methyltransferase
IFNAR
Ligand for E3 Ligase
PGE Synthase
Phospholipase
PLK
Tie-2
transporter
ACK1
CaMK
GluR
HSV
LDL
Molecular Glues
P2X Receptor
PROTACs
RIP kinase
SARS-CoV
Serine Protease
SGK
Sirtuin
Topoisomerase
TRP/TRPV Channel
Anti-infection
BACE
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
E1/E2/E3 Enzyme
Epigenetic Reader Domain
Estrogen/progestogen Receptor
Glucosidase
Glutathione Peroxidase
HBV
Hck
HSP
Immunology/Inflammation related
Integrin
IRAK
Ligands for Target Protein for PROTAC
Mitochondrial Metabolism
MRP
NADPH
NOD
p53
Pim
Transferase
Aryl Hydrocarbon Receptor
ATP Citrate Lyase
ATPase
BCRP
Beta-Secretase
Chloride channel
CRISPR/Cas9
FAAH
Fatty Acid Synthase
Gap Junction Protein
GPCR
GTPase
iGluR
IRE1
Leukotriene Receptor
Melanin-concentrating Hormone Receptor (MCHR)
MNK
Monoamine Transporter
Others
Proton pump
Reverse Transcriptase
Rho
ribosome
ROR
RSV
VDA
YAP
FOXO3
AAK1
AhR
Amylase
Androgen Receptor
Apelin receptor
Aromatase
Arrestin
cAMP
CFTR
Cholecystokinin Receptor
c-Myc
DAPK
Decarboxylase
DNA
DNA Alkylation
DNA Methyltransferase
DUB
Estrogen Receptor/ERR
FLAP
Free radical scavengers
FXR
Glucocorticoid Receptor
Glucokinase
GlyT
gp120/CD4
GRK
GST
Guanylate cyclase
Hedgehog/Smoothened
Hippo pathway
Histone Acetyltransferase
Histone Demethylase
Hydroxylase
IAP
Kinesin
LRRK2
LTR
Melatonin Receptor
MT Receptor
MyD88
Myosin
Na+/Ca2+ Exchanger
NADPH-oxidase
NMDAR
NOD-like Receptor (NLR)
NPC1L1
OCT
p97
PAD
PAI-1
PD-1/PD-L1
PERK
PKM
Progesterone Receptor
Protease
Pyroptosis
RAAS
RAR/RXR
Reductase
S1P Receptor
SGLT
Stearoyl-CoA Desaturase (SCD)
STING
Thrombopoietin Receptor
ADC Cytotoxin
Kras
TargetMol | Target Loading
正在加载 ~