抗结直肠癌化合物库

Anti-Colorectal Cancer Compound Library
产品编号: L2194

结直肠癌(Colorectal Cancer,CRC),又称大肠癌,包括结肠癌和直肠癌,是全球范围内致命的恶性肿瘤之一,严重威胁人类健康,近年来其发病率和死亡率均呈上升趋势,并且发病率随着年龄的增加而增加,人口老龄化和不良生活习惯是主要诱因,缺乏运动、肥胖、抽烟也使得患结直肠癌的风险显著增加。结直肠癌的治疗手段包括手术、放疗、化疗和靶向治疗。早期癌症可以通过手术治愈,晚期转移性癌通常选择化疗联合靶向治疗,研究表明,多个信号通路和靶点的失调与结直肠癌有关,如: VEGFR、EGFR、Wnt/β-catenin、p53、TGF-β等 TargetMol 抗结直肠癌化合物库收集了1880 种与结直肠癌相关的化合物,包括已经报道具有结直肠癌治疗作用的化合物,以及靶向结直肠癌相关靶点的化合物,是抗结直肠癌药物研发的良好工具。

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L2194
产品编号: L2194
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
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技术资料
产品描述
产品描述:
  • 1880种与结直肠癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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Apoptosis
Autophagy
PI3K
EGFR
VEGFR
COX
mTOR
p38 MAPK
Akt
ERK
Wnt/beta-catenin
AMPK
GSK-3
Raf
NF-κB
c-Met/HGFR
CDK
PDGFR
STAT
MAPK
JNK
Ras
TGF-beta/Smad
MEK
p53
c-Kit
Src
FGFR
FLT
Antibacterial
Endogenous Metabolite
DNA-PK
DNA/RNA Synthesis
S6 Kinase
ATM/ATR
HER
ALK
Mdm2
Parasite
PDK
c-RET
TNF
PKC
Reactive Oxygen Species
Gamma-secretase
JAK
Aurora Kinase
Antibiotic
Potassium Channel
Ferroptosis
Caspase
E1/E2/E3 Enzyme
Bcr-Abl
Kras
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PKA
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IGF-1R
PI4K
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PPAR
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Influenza Virus
Tyrosine Kinases
IL Receptor
TAM Receptor
Lipoxygenase
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HIV Protease
Calcium Channel
Topoisomerase
MMP
Bcl-2 Family
FAK
Cytochromes P450
MNK
Trk receptor
Sirtuin
HDAC
MLK
NOS
Others
Antioxidant
Phosphatase
ROCK
Chk
Prostaglandin Receptor
Beta Amyloid
Nucleoside Antimetabolite/Analog
SIK
PDE
Epigenetic Reader Domain
Sodium Channel
HCV Protease
ROS
HSV
PTEN
Antiviral
IκB/IKK
Microtubule Associated
Carbonic Anhydrase
Virus Protease
HSP
TLR
MELK
Syk
Tyrosinase
NO Synthase
DYRK
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TOPK
Adrenergic Receptor
Aryl Hydrocarbon Receptor
IAP
Drug Metabolite
Interleukin
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Ephrin Receptor
ASK
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Phospholipase
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GTPase
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LDL
Mitochondrial Metabolism
Glucosidase
DNA Alkylation
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PGE Synthase
P-gp
GABA Receptor
5-HT Receptor
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HIF/HIF Prolyl-Hydroxylase
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transporter
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IRE1
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cAMP
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Discoidin Domain Receptor (DDR)
Gap Junction Protein
BMI-1
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Kinesin
Apelin receptor
MicroRNA
NPC1L1
RAR/RXR
DHFR
Dopamine Receptor
ROR
Amino Acids and Derivatives
MyD88
Ligands for Target Protein for PROTAC
YAP
Arginase
Reductase
RAAS
PERK
Progesterone Receptor
OCT
c-Myc
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Hck
Neurotensin Receptor
Leukotriene Receptor
FXR
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iGluR
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MTH1
Opioid Receptor
Fatty Acid Synthase
Somatostatin
KSP
DNA
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Androgen Receptor
ATP Citrate Lyase
Wee1
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CD73
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hCE
PAI-1
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Hippo pathway
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RXFP receptor
DAPK
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NOD
Protease-activated Receptor
AhR
PD-1/PD-L1
S1P Receptor
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