抗结直肠癌化合物库

Anti-Colorectal Cancer Compound Library
产品编号: L2194

结直肠癌(Colorectal Cancer,CRC),又称大肠癌,包括结肠癌和直肠癌,是全球范围内致命的恶性肿瘤之一,严重威胁人类健康,近年来其发病率和死亡率均呈上升趋势,并且发病率随着年龄的增加而增加,人口老龄化和不良生活习惯是主要诱因,缺乏运动、肥胖、抽烟也使得患结直肠癌的风险显著增加。结直肠癌的治疗手段包括手术、放疗、化疗和靶向治疗。早期癌症可以通过手术治愈,晚期转移性癌通常选择化疗联合靶向治疗,研究表明,多个信号通路和靶点的失调与结直肠癌有关,如: VEGFR、EGFR、Wnt/β-catenin、p53、TGF-β等 TargetMol 抗结直肠癌化合物库收集了1880 种与结直肠癌相关的化合物,包括已经报道具有结直肠癌治疗作用的化合物,以及靶向结直肠癌相关靶点的化合物,是抗结直肠癌药物研发的良好工具。

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L2194
产品编号: L2194
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
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技术资料
产品描述
产品描述:
  • 1880种与结直肠癌相关的化合物,可以用于高通量和高内涵筛选;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库组成
Apoptosis
Autophagy
PI3K
EGFR
VEGFR
COX
mTOR
p38 MAPK
Akt
ERK
AMPK
Wnt/beta-catenin
GSK-3
Raf
NF-κB
c-Met/HGFR
CDK
PDGFR
STAT
MAPK
JNK
Ras
TGF-beta/Smad
MEK
p53
c-Kit
Src
FGFR
Antibacterial
FLT
Endogenous Metabolite
DNA-PK
S6 Kinase
DNA/RNA Synthesis
ATM/ATR
HER
ALK
Parasite
Mdm2
PDK
c-RET
TNF
PKC
Reactive Oxygen Species
Gamma-secretase
Antibiotic
Aurora Kinase
Caspase
JAK
Potassium Channel
Bcr-Abl
E1/E2/E3 Enzyme
Ferroptosis
PARP
Kras
Antifungal
IGF-1R
Mitophagy
PKA
PI4K
Rho
Casein Kinase
Dehydrogenase
Influenza Virus
PPAR
IL Receptor
TAM Receptor
Tyrosine Kinases
Bcl-2 Family
c-Fms
Lipoxygenase
Calcium Channel
Cytochromes P450
FAK
HIV Protease
Trk receptor
HDAC
MLK
MMP
MNK
Sirtuin
Topoisomerase
Antioxidant
Beta Amyloid
Chk
NOS
Others
Phosphatase
Prostaglandin Receptor
ROCK
Epigenetic Reader Domain
PDE
SIK
Sodium Channel
Antiviral
HCV Protease
HSV
IκB/IKK
Microtubule Associated
Nucleoside Antimetabolite/Analog
PTEN
ROS
Carbonic Anhydrase
HSP
MELK
NO Synthase
Syk
TLR
Virus Protease
AChR
Adrenergic Receptor
Aryl Hydrocarbon Receptor
ASK
Drug Metabolite
DYRK
Ephrin Receptor
IAP
Interleukin
Nrf2
Phospholipase
Porcupine
ROS Kinase
SGK
Tie-2
TOPK
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5-HT Receptor
DNA Alkylation
Estrogen/progestogen Receptor
GABA Receptor
Glucosidase
GTPase
HIF
HIF/HIF Prolyl-Hydroxylase
Hydroxylase
Integrin
LDL
Mitochondrial Metabolism
PGE Synthase
P-gp
RIP kinase
Serine Protease
TRP/TRPV Channel
BTK
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ATPase
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CSF-1R
DNA Alkylator/Crosslinker
Estrogen Receptor/ERR
GluR
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GPCR
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IRAK
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transporter
ACK1
ADC Cytotoxin
Adenosine Receptor
APC/C
BACE
Beta-Secretase
BMI-1
CaMK
cAMP
Cannabinoid Receptor
CCR
Chloride channel
Discoidin Domain Receptor (DDR)
DNA Methyltransferase
FAAH
Gap Junction Protein
HBV
Histamine Receptor
IRE1
Kinesin
LRRK2
NMDAR
PROTACs
Proton pump
RSV
SARS-CoV
Serine/threonin kinase
Transferase
Acyltransferase
AhR
Amino Acids and Derivatives
Androgen Receptor
Apelin receptor
Arginase
Aromatase
ATP Citrate Lyase
BCRP
CD73
Cholecystokinin Receptor
c-Myc
CRISPR/Cas9
DAPK
Decarboxylase
DHFR
DNA
Dopamine Receptor
DUB
Fatty Acid Synthase
FLAP
FXR
Glucocorticoid Receptor
Glucokinase
GPX
hCE
Hck
Hippo pathway
Histone Acetyltransferase
iGluR
KSP
Leukotriene Receptor
Ligands for Target Protein for PROTAC
Methionine Adenosyltransferase (MAT)
MicroRNA
MTH1
MyD88
Myosin
NADPH-oxidase
Neurotensin Receptor
NOD
NPC1L1
OCT
Opioid Receptor
PAI-1
PD-1/PD-L1
PERK
Progesterone Receptor
Protease-activated Receptor
RAAS
RAR/RXR
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Retinoid Receptor
Reverse Transcriptase
ROR
RXFP receptor
S1P Receptor
Somatostatin
UGT
Wee1
YAP
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