抗结直肠癌中药单体化合物库

Anti-Colorectal Cancer Traditional Chinese Medicine Compound Library
产品编号: L6740

结直肠癌(Colorectal Cancer,CRC)是常见的恶性肿瘤之一。大部分结直肠癌的病例是散发性的,由于目前的饮食习惯和生活方式,包括大量肉类、酒精和缺乏足够的体育锻炼,结直肠癌的发病率在全球范围内呈上升趋势。结直肠癌具有发病隐匿,预后差的特点,因此对其有效预防和干预策略存在强烈的公共卫生需求。
随着结直肠癌发病机制研究的日渐深入,中药有效成分在预防和治疗结肠癌方面的应用也得到了深入研究。中药可以通过调节多种信号通路,参与调节癌细胞的增殖、分化和凋亡,破坏癌细胞的生存环境,增强机体免疫系统,从而抑制结直肠癌的发生和发展。
TargetMol 抗结直肠癌中药单体化合物库,精选382 种抗结直肠癌相关的中药单体成分,来源包含补益类(如人参、黄芪)和清热解毒类(如黄芩、大黄)等多种中药成分,具有较为明确的生物活性信息,为抗结直肠癌相关研究提供有力工具。

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L6740
产品编号: L6740
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品描述:
  • 382种抗结直肠癌相关的中药单体集合,是药物开发、药理研究的有效工具;
  • 结构多样,包含黄酮、皂苷、萜类、生物碱等类别;
  • 靶向Wnt/beta-catenin、TGF-beta/Smad、NF-κB、Notch等多种靶点;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
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化合物库咨询
验证码
化合物库组成
Apoptosis
Autophagy
NF-κB
COX
p38 MAPK
Endogenous Metabolite
ERK
Akt
STAT
Antibacterial
AMPK
PI3K
Reactive Oxygen Species
JNK
Caspase
TNF
Others
EGFR
Parasite
IL Receptor
PARP
Wnt/beta-catenin
Antifungal
Bcl-2 Family
HIV Protease
Influenza Virus
PPAR
TGF-beta/Smad
Antioxidant
Cytochromes P450
Nrf2
Ferroptosis
mTOR
NO Synthase
NOS
Topoisomerase
DNA/RNA Synthesis
Lipoxygenase
MEK
Mitophagy
p53
Antibiotic
JAK
MMP
P-gp
Prostaglandin Receptor
ROS
Virus Protease
Antifection
ATPase
Cholinesterase (ChE)
Gamma-secretase
GSK-3
MAPK
PKC
TLR
Tyrosinase
VEGFR
Anti-infection
Beta Amyloid
CDK
Estrogen Receptor/ERR
Estrogen/progestogen Receptor
HCV Protease
HIF
HIF/HIF Prolyl-Hydroxylase
Integrin
Potassium Channel
PTEN
5-HT Receptor
c-Met/HGFR
FGFR
GABA Receptor
HSV
IGF-1R
Interleukin
IκB/IKK
Mitochondrial Metabolism
PDE
Phospholipase
S6 Kinase
Sirtuin
transporter
AChR
Antiviral
Calcium Channel
CXCR
Dehydrogenase
Epigenetic Reader Domain
FAK
Glucosidase
HBV
HDAC
HER
IAP
LDL
MAO
NOD
Proton pump
Ras
Retinoid Receptor
SARS-CoV
TRP/TRPV Channel
UGT
ADC Cytotoxin
Adenosine Receptor
Adrenergic Receptor
ALK
Aminopeptidase
Aromatase
ATM/ATR
BACE
Bcr-Abl
Beta-Secretase
cAMP
Carbonic Anhydrase
CCR
c-Myc
E1/E2/E3 Enzyme
FAAH
Fatty Acid Synthase
Glucokinase
gp120/CD4
GPCR
hCE
Histone Acetyltransferase
Immunology/Inflammation related
Lipase
MicroRNA
Monoamine Oxidase
MRP
NADPH
NMDAR
NOD-like Receptor (NLR)
NPC1L1
OCT
Opioid Receptor
PAFR
PAI-1
PD-1/PD-L1
PDK
PERK
PGE Synthase
Phosphatase
PKA
RAAS
Raf
RAR/RXR
Reverse Transcriptase
ROS Kinase
RSV
Sodium Channel
Survivin
Transferase
Xanthine Oxidase
化合物库信息示例
Empty989-51-596087-21-7957-66-494805-82-094-41-791653-50-888930-15-888495-63-0882664-74-6874485-32-2Empty
(-)-Epigallocatechin GallateStylopine hydrochlorideIsolinderalactoneGlycycoumarinChalconeZingiberen newsaponinMogrolArtesunatePolygalasaponin F25(R,S)-Ruscogenin
Empty87205-99-0855-97-085026-55-784745-95-984709-25-184687-43-484680-75-184676-89-184-26-483-79-4Empty
Dihydrotanshinone I5,7,3',4'-TetramethoxyflavoneRosinEriocalyxin Bd-EpigalbacinAstragaloside IVAstragaloside IAstragaloside IIRutaecarpineRotenone
Empty83-46-5831-61-882854-37-382508-31-482-02-081907-62-280681-45-480418-24-280321-69-378281-02-4Empty
Beta-SitosterolEthyl gallateEchinacosidePseudolaric Acid BKhellinGanoderic acid APrim-O-glucosylcimifuginNotoginsenoside R1Gypenoside XVIIHydroxysafflor yellow A
Empty78214-33-277-59-8775351-88-777-52-17689-03-476822-21-476-66-476474-56-176376-43-776296-75-8Empty
Ginsenoside Rh2TomatidineCorylifol AUrsolic acidCamptothecinDanshensuRhynchophyllineDihydrocurcuminEuphorbia factor L1Polyphyllin G
Empty761425-93-875887-54-6751-03-174805-91-7735-46-673255-40-073069-25-773069-14-473030-71-471835-85-3Empty
Clematichinenoside ARArtemotilObacunoneMethylophiopogonanone BHamaudolMoringin(±)-Praeruptorin AAtractylenolide IIAtractylenolide IIIPhenethyl ferulate
Empty70831-56-06882-68-46877-32-36873-13-86873-09-268370-47-868124-04-96807-83-667979-25-367884-30-4Empty
L-Chicoric AcidSophoridineCorynoxinePhellodendrineEpiberberineMicheliolideParis saponin VIITrifolirhizinAurantio-obtusinDendrobium phenol
Empty66656-92-666648-50-866648-44-06601-66-765914-17-265-45-2652-78-86483-15-4642-38-663968-64-9Empty
Esculentoside HEthyl trans-caffeateN-​Feruloyloctopamine6-Demethoxytangeretin(E/Z)-PolydatinSalicylamideGossypinSophocarpineL-quebrachitolArtemisinin
Empty632-85-963223-86-963177-57-1630-94-462596-29-6623-05-262014-87-36199-67-36192-62-761521-74-2Empty
WogoninGinsenoside Rh1Methyl 2,5-dihydroxycinnamateCorynoxeineMorusin4-Hydroxybenzyl alcoholHelichrysetinCucurbitacin BTOMATIDINE HYDROCHLORIDE(+)-Nortrachelogenin
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