抗乳腺癌化合物库

Anti-Breast Cancer Compound Library
产品编号: L2191

乳腺癌是乳腺恶性肿瘤,是全球女性发病率较高的癌症,约占女性癌症患者的20%,也是100多个国家癌症死亡的主要原因。近年来全球乳腺癌发病率一直呈上升趋势。 乳腺癌根据病理分型可分为非浸润性癌,早期浸润性癌,浸润性癌。根据分子分型可分为雌激素受体阳性乳腺癌(ER+PR+HER2-),HER2阳性乳腺癌(ER-PR-HER2+),三阴性乳腺癌(ER-PR-HER2-)。不同类型的乳腺癌,从治疗方法到预后都是非常不同,需要针对已经明确的致癌位点,探索相关靶点来设计相应的药物。 TargetMol 抗乳腺癌库收集了2440 种与乳腺癌相关的化合物,包含了已经报道的有乳腺癌治疗作用的化合物,以及相关的靶点通路(HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA 等),是乳腺癌药物研发的良好工具。

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L2191
产品编号: L2191
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品描述:
  • 2440种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
  • 靶点包含HER-2, VEGF, EGFR, PARP, CDK4/6, HSP, PD-1, SET7/9, BRCA等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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Apoptosis
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NF-κB
PI3K
CDK
EGFR
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VEGFR
COX
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transporter
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ABC Transporter
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Gap Junction Protein
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化合物库信息示例
Empty99873-43-599-66-199-32-199-24-199105-77-8989-51-598619-25-1978-62-197682-44-597-53-0Empty
DroxinostatValproic AcidChelidonic acidMethyl gallateSulcotrione(-)-Epigallocatechin GallateSchisandroneIMD-0354IrinotecanEugenol
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TroglitazoneMomordin Ic2-hexyl-4-Pentynoic Acid(E)-Akt inhibitor-IVGuggulsteroneNIH-128484'-MethoxychalconeGSK1059615IpsapironeDPA-714
Empty957-68-6957054-33-0957054-30-7956958-53-5955977-50-1955900-27-3955365-80-7952021-60-2951151-97-6950762-95-5Empty
7-Aminocephalosporanic acidPictilisib dimethanesulfonatePictilisibPilaralisib analoguePI-3065RK-9123016AdavosertibPF 477736JNJ-38158471PCI-34051
Empty95058-81-494987-08-394805-82-0946518-60-1945619-74-9945189-68-4944396-88-7944396-07-0944328-88-594-41-7Empty
GemcitabineGypenoside XLIXGlycycoumarinLY2409881 trihydrochlorideOPHIOPOGONIN DSJ000063181NIBR-17BuparlisibQS11Chalcone
Empty943820-93-7943319-70-8943119-42-4942918-07-2942655-44-9942425-68-5942289-87-4941575-71-9939791-38-5938-55-6Empty
Wnt/β-catenin agonist 2PonatinibOUL232GSK-1070916JK-P3PHA-767491 hydrochloridePI-828BIP-135PF-562271 besylate6-(Dimethylamino)purine
Empty938440-64-393772-31-7937265-83-3937263-43-9937174-76-0937039-45-7936890-98-1936446-61-6936345-35-6936345-34-5Empty
KU-0063794Neogambogic acidARRY-380 (analog )TucatinibGSK-690693Pimelic diphenylamide 106OSI-027NRC-2694PF-02413873Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl-
Empty935881-37-1934828-12-3934826-68-3934541-31-8934526-89-3934493-76-2934389-88-5934353-76-1934343-74-5934162-61-5Empty
AR42CXD101VisomitinTAK-901PilaralisibVoxtalisibLY-294002 hydrochlorideENMD-2076NVP-HSP990A-966492
Empty932359-76-7931417-26-493117-08-993-07-2930039-92-2929016-96-692831-11-3928037-13-2927961-18-0927885-00-5Empty
FiVe1ANI-75-AIQVeratric acidBRD4 Inhibitor-27PracinostatMN-64GolvatinibLanifibranorHS-1793
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