尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。 根据文献报道和有关公开资料,我们挑选了 3970 个具有已知抗癌活性的化合物组成抗癌活性库,可用于具体癌症的阳性对照及癌症机理的研究。希望我们在抗癌研究的路上,助您一臂之力!
Empty | 99-66-1 | 99614-01-4 | 99-24-1 | 99011-78-6 | 99011-02-6 | 99009-20-8 | 989-51-5 | 989-30-0 | 989-23-1 | 98891-44-2 | Empty |
Valproic Acid | Ondansetron hydrochloride | Methyl gallate | Imiquimod hydrochloride | Imiquimod | Pyrazoloacridine | (-)-Epigallocatechin Gallate | 3-Epiursolic acid | Deoxylimonin | Pseudolaric acid A-O-β-D-glucopyranoside | ||
Empty | 987-65-5 | 98665-15-7 | 98474-78-3 | 97938-30-2 | 97919-22-7 | 97682-44-5 | 97-65-4 | 97322-87-7 | 97230-47-2 | 97230-46-1 | Empty |
ATP disodium salt | Ganoderic acid F | Pseudoginsenoside RT5 | Sophoraflavanone G | Chloroquinoxaline sulfonamide | Irinotecan | Itaconic acid | Troglitazone | Picfeltarraenin IA | Picfeltarraenin IB | ||
Empty | 97207-47-1 | 97-18-7 | 970-74-1 | 970-73-0 | 96990-18-0 | 965-52-6 | 96187-53-0 | 961-29-5 | 960374-59-8 | 96020-91-6 | Empty |
Meisoindigo | Bithionol | (-)-Epigallocatechin | (+)-Gallocatechin | Momordin Ic | Nifuroxazide | Brequinar | Isoliquiritigenin | ONX-0914 | Eflornithine hydrochloride hydrate | ||
Empty | 959-23-9 | 95923-66-3 | 958852-01-2 | 958843-91-9 | 95847-70-4 | 958233-07-3 | 958-09-8 | 95809-78-2 | 957-77-7 | 957-66-4 | Empty |
4'-Methoxychalcone | YM 534 | GSK1059615 | CMLD-2 | Ipsapirone | DPA-714 | 2'-Deoxyadenosine | Devimistat | 5-Hydroxyuridine | Isolinderalactone | ||
Empty | 957054-33-0 | 957054-30-7 | 956958-53-5 | 956905-27-4 | 956697-53-3 | 956590-23-1 | 956154-63-5 | 956104-40-8 | 955900-27-3 | 955365-80-7 | Empty |
Pictilisib dimethanesulfonate | Pictilisib | Pilaralisib analogue | PF-04217903 | Sonidegib | UNBS5162 | TCS HDAC6 20b | Apalutamide | RK-9123016 | Adavosertib | ||
Empty | 953769-46-5 | 95311-94-7 | 95258-14-3 | 952021-60-2 | 951-77-9 | 95104-27-1 | 950-99-2 | 950769-58-1 | 950762-95-5 | 95058-81-4 | Empty |
Sotuletinib | Lucideric acid A | Yadanziolide A | PF 477736 | 2'-Deoxycytidine | Tetrazolast | 2,2,5,7,8-Pentamethyl-6-Chromanol | Quizartinib | PCI-34051 | Gemcitabine | ||
Empty | 95041-90-0 | 948557-43-5 | 94705-70-1 | 946150-57-8 | 946128-88-7 | 945923-91-1 | 945771-74-4 | 945595-80-2 | 94497-51-5 | 944547-46-0 | Empty |
Erianin | Tie2 kinase inhibitor 1 | Gypenoside XLVI | Remetinostat | Ro 5126766 | Fmoc-1,6-diaminohexane hydrochloride | BNC105 | AMG 900 | Tamibarotene | Mycro 3 | ||
Empty | 944396-07-0 | 944328-88-5 | 944261-79-4 | 94-41-7 | 943820-93-7 | 94356-22-6 | 943540-75-8 | 943540-74-7 | 943332-08-9 | 943319-70-8 | Empty |
Buparlisib | QS11 | A-803467 | Chalcone | Wnt/β-catenin agonist 2 | Rhapontigenin 3'-O-glucoside | JNJ-38877605 | JNJ-38877618 | Selumetinib sulfate | Ponatinib |