抗心血管疾病化合物库

Anti-Cardiovascular Disease Compound Library
产品编号: L5400

心血管疾病泛指由于动脉粥样硬化、高脂血症、血液黏稠、高血压等所导致的心脏、大脑及全身组织发生的缺血性或出血性疾病,例如心绞痛、心肌梗塞、中风等,是全球死亡的首要原因。不同类型疾病的发病机制不同,各种抗氧化、抗高血脂、抗缺血、抑制血小板聚集和抗炎物质都具有降低心血管疾病风险的作用。某些天然产物具有抑制粘附分子、细胞因子和趋化因子基因表达,抑制血小板功能,增强内皮细胞一氧化氮释放,抑制平滑肌活化的作用,这些化合物都是心血管疾病药物筛选中的重要工具。 TargetMol 抗心血管疾病化合物库是由 1793 个心血管疾病相关的化合物组成的综合筛选库,用于心血管疾病的相关研究和高通量高内涵筛选。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L5400
产品编号: L5400
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品描述:
  • 1793种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括膜转运体、离子通道等心血管疾病相关靶点;
  • 大部分产品是经FDA、EMA或NMPA批准上市的药物,是研究心血管相关疾病的有效工具;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
我们的化合物库可以灵活定制! 了解更多
化合物库咨询
验证码
化合物库组成
Adrenergic Receptor
Calcium Channel
PDE
Apoptosis
Autophagy
VEGFR
Others
COX
Sodium Channel
Endogenous Metabolite
Potassium Channel
5-HT Receptor
AChR
RAAS
PDGFR
Dopamine Receptor
Antibacterial
TNF
NF-κB
IL Receptor
Histone Acetyltransferase
FGFR
PARP
Histamine Receptor
FLT
c-Kit
PPAR
Parasite
CDK
PKC
HMG-CoA Reductase
BACE
Factor Xa
Reactive Oxygen Species
EGFR
Antioxidant
Adenosine Receptor
Epigenetic Reader Domain
Carbonic Anhydrase
JAK
IGF-1R
Cytochromes P450
ATPase
Antifungal
Antibiotic
Src
p38 MAPK
c-Met/HGFR
Mitophagy
Influenza Virus
c-RET
Thrombin
TRP/TRPV Channel
Norepinephrine
Ferroptosis
Phospholipase
P2Y Receptor
ERK
Glucocorticoid Receptor
Lipoxygenase
Beta-Secretase
HIV Protease
PI3K
Drug Metabolite
Akt
DNA/RNA Synthesis
PKA
ROS
P-gp
Prostaglandin Receptor
Beta Amyloid
HER
NO Synthase
MRP
Raf
Guanylate cyclase
CaMK
Nrf2
STAT
HDAC
GABA Receptor
Proteasome
GSK-3
iGluR
Bcr-Abl
NMDAR
Aurora Kinase
Interleukin
SARS-CoV
Acetyl-CoA Carboxylase
Proton pump
Integrin
Dehydrogenase
CETP
Virus Protease
Tyrosine Kinases
Serotonin Transporter
Serine/threonin kinase
ROCK
Topoisomerase
Mitochondrial Metabolism
Angiotensin-converting Enzyme (ACE)
c-Fms
AMPK
Hydroxylase
MEK
Anti-infection
NOD
Chloride channel
Serine Protease
Liver X Receptor
Caspase
MAO
P2X Receptor
GluR
Acyltransferase
Trk receptor
IκB/IKK
Tyrosinase
HIF/HIF Prolyl-Hydroxylase
NOS
NADPH
Tie-2
Glutathione Peroxidase
Wnt/beta-catenin
Nucleoside Antimetabolite/Analog
LDL
Opioid Receptor
DPP-4
HSV
Cholinesterase (ChE)
Chk
Epoxide Hydrolase
cAMP
PGE Synthase
Ephrin Receptor
Neprilysin
HIF
Sigma receptor
TAM Receptor
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
p53
Monoamine Oxidase
Thyroid hormone receptor(THR)
Estrogen/progestogen Receptor
Arginase
DNA Alkylator/Crosslinker
JNK
Antifolate
FXR
CSF-1R
Myosin
Na-K-Cl cotransporter
HCN Channel
Fatty Acid Synthase
Endothelin Receptor
mTOR
TLR
Bcl-2 Family
transporter
RSV
Reverse Transcriptase
PDK
Platelet aggregation
Syk
NADPH-oxidase
S6 Kinase
Microtubule Associated
FAK
Adenylyl Cyclase
Transferase
DHFR
Histone Methyltransferase
Amino Acids and Derivatives
LTR
Na+/Ca2+ Exchanger
Histone Demethylase
Estrogen Receptor/ERR
HBV
Rho
Leukotriene Receptor
PYK2
Amylase
Immunology/Inflammation related
UGT
PAFR
ABC Transporter
Antifection
Monoamine Transporter
DNA Alkylation
FAAH
Xanthine Oxidase
DNA
Androgen Receptor
TGF-beta/Smad
MAPK
Aminopeptidase
Sirtuin
PAI-1
ALK
GST
GPR
SGK
DNA Methyltransferase
AhR
NPC1L1
Monocarboxylate transporter
ROR
DNA-PK
HCV Protease
DprE1
YAP
Reductase
IFNAR
Lipase
PERK
Phosphatase
Progesterone Receptor
N-Acetylglucosaminyltransferase
VDAC
Cell Cycle Arrest
Cysteine Protease
Neurotensin Receptor
Glucokinase
Aryl Hydrocarbon Receptor
IAP
IRE1
Annexin A
FLAP
RIP kinase
Adiponectin Receptor
GRK
DNA gyrase
GlyT
Glucosidase
Anion Exchanger
Isocitrate Dehydrogenase (IDH)
CCR
ACK1
Vasopressin Receptor
MMP
Thrombopoietin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
Lipid
BCRP
OAT
Antiviral
HSP
Decarboxylase
ASK
Casein Kinase
Retinoid Receptor
Aromatase
CRISPR/Cas9
RXFP receptor
PLK
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
Gap Junction Protein
IRAK
Ras
p97
CFTR
MLK
PKM
S1P Receptor
ADC Cytotoxin
Sodium-dependent phosphate transporter
Vitamin
BTK
TargetMol | Target Loading
正在加载 ~