抗纤维化化合物库

Anti-Fibrosis Compound Library
产品编号: L9810

纤维化(fibrosis)是一种病理改变,主要表现为器官组织内纤维结缔组织增多,实质细胞减少,持续进展可致器官结构破坏和功能减退,乃至衰竭,严重威胁人类健康和生命。纤维化可发生于多种器官,常见的包括肺脏、肝脏、肾脏、骨髓等。纤维化通常由各种刺激导致的慢性炎症性反应引起,包括:持续性感染,自身免疫反应,过敏性反应,化学刺激,射线和组织损伤等。

TargetMol 抗纤维化化合物库收集了1800 种抗纤维化分子和潜在的抗纤维化分子,包括相关靶点如TGFβ、TNFα、MMP 的抑制剂、抗氧化剂及抗炎分子等,是研究纤维化机制和开发抗纤维化药物的良好工具。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L9810
产品编号: L9810
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品特性:
  • 1800种潜在的抗纤维化分子,是研究纤维化的有效工具,可以用于高通量筛选和高内涵筛选;
  • 靶点包括TGFβ、TNFα、MMP、EGFR、NADPH-oxidase等;
  • 部分化合物已经得到FDA批准上市;?
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库信息示例
Empty99697-24-299464-64-999353-00-199-32-199-24-1989-51-5978-62-197-53-0973-67-1970-74-1Empty
24-Norursodeoxycholic acidAmpiroxicamMethyl rosmarinateChelidonic acidMethyl gallate(-)-Epigallocatechin GallateIMD-0354Eugenol5,6,7-TRIMETHOXYFLAVONE(-)-Epigallocatechin
Empty96990-18-096574-01-596087-21-7959841-49-795975-55-6959551-10-1958941-60-1958852-01-2957054-33-0957054-30-7Empty
Momordin IcSalvianolic acid AStylopine hydrochloride(E)-Akt inhibitor-IVGuggulsteroneNIH-12848CFTR corrector 12GSK1059615Pictilisib dimethanesulfonatePictilisib
Empty956958-53-5955977-50-195311-94-7952021-60-2950736-05-794805-82-0946518-60-1946128-88-7946002-48-8945755-56-6Empty
Pilaralisib analoguePI-3065Lucideric acid APF 477736B-Raf IN 1GlycycoumarinLY2409881 trihydrochlorideRo 5126766SAG 21kXL019
Empty945619-74-9945614-12-0945595-80-2945189-68-494492-24-7944396-07-0943820-93-7943764-99-6943319-70-8942918-07-2Empty
OPHIOPOGONIN DPexmetinibAMG 900SJ0000631812'-acetylacteosideBuparlisibWnt/β-catenin agonist 2AcebilustatPonatinibGSK-1070916
Empty942655-44-9942507-42-8942425-68-5942183-80-4941685-37-6941678-49-594055-76-2940310-85-0938440-64-3937807-66-4Empty
JK-P3AZ304PHA-767491 hydrochlorideSCH772984Ruxolitinib (S enantiomer)RuxolitinibSuplatast (Tosilate)NVP-BHG712KU-0063794Neurodazine
Empty937272-79-2937174-76-0936890-98-1936727-05-8936091-26-8935273-79-3934826-68-3934660-93-2934541-31-8934526-89-3Empty
PacritinibGSK-690693OSI-027LumacaftorFedratinibMK-4101VisomitinCobimetinibTAK-901Pilaralisib
Empty934493-76-2934389-88-5934353-76-193-35-6931706-15-9931695-79-393-07-2929007-72-7928037-13-2927880-90-8Empty
VoxtalisibLY-294002 hydrochlorideENMD-2076UmbelliferonePPQ-102ML-191Veratric acidDB07268GolvatinibRAF265
Empty925705-73-3925701-49-1923564-51-6923032-37-5919936-70-2918505-84-7918505-61-0918504-65-1917111-44-5916232-21-8Empty
TG 100713KU60019NavitoclaxRefametinibGS87PLX-4720BRAF inhibitorVemurafenibLexibulinGS143
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