抗胰腺癌化合物库

Anti-Pancreatic Cancer Compound Library
产品编号: L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。 为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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L2192
产品编号: L2192
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品特点:
  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库组成
Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
PPAR
Wnt/beta-catenin
mTOR
Akt
JAK
HDAC
PARP
STAT
Src
GSK-3
ERK
AMPK
FGFR
p38 MAPK
Endogenous Metabolite
Antibacterial
c-Met/HGFR
Raf
PDGFR
FLT
HER
TGF-beta/Smad
p53
c-Kit
MEK
JNK
MMP
Reactive Oxygen Species
IGF-1R
TNF
Parasite
Ras
Caspase
Bcr-Abl
DNA-PK
S6 Kinase
Tyrosine Kinases
ATM/ATR
Aurora Kinase
ALK
MAPK
IL Receptor
HIF/HIF Prolyl-Hydroxylase
Cytochromes P450
DNA/RNA Synthesis
Potassium Channel
Antibiotic
Mdm2
Ferroptosis
PDK
c-RET
Pim
Gamma-secretase
STING
Influenza Virus
HIV Protease
Mitophagy
HIF
Hedgehog/Smoothened
E1/E2/E3 Enzyme
Bcl-2 Family
Kras
Antifungal
PKC
Lipoxygenase
PD-1/PD-L1
PKA
Calcium Channel
PI4K
Dehydrogenase
Casein Kinase
FAK
NO Synthase
Prostaglandin Receptor
Nrf2
Trk receptor
IκB/IKK
NOS
Virus Protease
Topoisomerase
Chk
Epigenetic Reader Domain
Interleukin
Beta Amyloid
Rho
PDE
ROS
c-Fms
Tyrosinase
Sirtuin
TAM Receptor
HCV Protease
Phosphatase
HSV
Antioxidant
ROCK
PTEN
P-gp
5-HT Receptor
AChR
Sodium Channel
Others
DYRK
Adrenergic Receptor
SIK
Mitochondrial Metabolism
Antifection
PGE Synthase
GABA Receptor
Syk
Microtubule Associated
Proteasome
ATPase
Estrogen/progestogen Receptor
Adenosine Receptor
Tie-2
Aryl Hydrocarbon Receptor
CSF-1R
Drug Metabolite
Smo
Antiviral
TLR
Ephrin Receptor
PLK
Anti-infection
Carbonic Anhydrase
Integrin
TRP/TRPV Channel
IAP
RIP kinase
HSP
transporter
MELK
GPR
SGK
IRAK
MLK
BTK
Chloride channel
IFNAR
PERK
Histamine Receptor
GTPase
c-Myc
Estrogen Receptor/ERR
HBV
Cholecystokinin Receptor
Hck
Serine Protease
Serine/threonin kinase
PYK2
LDL
Glucosidase
CCR
Cholinesterase (ChE)
Cannabinoid Receptor
ROS Kinase
Transferase
Histone Methyltransferase
DNA Alkylator/Crosslinker
BACE
NADPH
RAAS
Glutathione Peroxidase
MRP
Nucleoside Antimetabolite/Analog
Leukotriene Receptor
Glucocorticoid Receptor
Immunology/Inflammation related
NMDAR
Opioid Receptor
DNA Alkylation
cAMP
CaMK
DUB
Androgen Receptor
Acyltransferase
Porcupine
SARS-CoV
LRRK2
Free radical scavengers
Decarboxylase
Retinoid Receptor
Phospholipase
Discoidin Domain Receptor (DDR)
NOD
NOD-like Receptor (NLR)
Proton pump
Dopamine Receptor
ADC Cytotoxin
Histone Demethylase
Progesterone Receptor
Cell Cycle Arrest
Glucokinase
UGT
ABC Transporter
FAAH
ACK1
GluR
ATP Citrate Lyase
Lipid
Beta-Secretase
MNK
Histone Acetyltransferase
Pyroptosis
RSV
Reverse Transcriptase
Aromatase
Gap Junction Protein
NADPH-oxidase
S1P Receptor
Melanin-concentrating Hormone Receptor (MCHR)
Adenylyl Cyclase
MicroRNA
NPC1L1
RAR/RXR
DHFR
ROR
YAP
Arginase
LPL Receptor
LTR
Na+/Ca2+ Exchanger
Reductase
gp120/CD4
TOPK
VDA
OCT
Liver X Receptor
Cysteine Protease
FXR
iGluR
Myosin
IRE1
FLAP
PAFR
Haspin Kinase
Monoamine Transporter
Hexokinase
Guanylate cyclase
DPP-4
Fatty Acid Synthase
Thioredoxin
PAK
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
DNA
BCRP
Aminopeptidase
ASK
hCE
PAI-1
Methionine Adenosyltransferase (MAT)
Hippo pathway
LPA Receptor
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
DAPK
BMI-1
DNA Methyltransferase
Sigma receptor
Thrombin
p97
CFTR
Kinesin
PKM
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