抗胰腺癌化合物库

Anti-Pancreatic Cancer Compound Library
产品编号: L2192

随着医学技术的进步,大部分癌症的生存率都在提高,例如乳腺癌,结直肠癌等肿瘤,近几十年来,生存率得到了大幅度的提升。但是,有一个例外,那就是胰腺癌,胰腺癌是一种发病隐匿,进展迅速,治疗效果和预后极差的消化道恶性肿瘤。胰腺癌的生存率一直停滞不前,胰腺癌的五年生存率只有5%至10%,绝大部分患者在诊断胰腺癌半年内死亡,由于生存率低,死亡率高,胰腺癌称为癌中之王。 为了满足胰腺癌研究客户的需求,TargeMol 收集了 2508 种与胰腺癌相关的化合物,作用于 KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等胰腺癌相关靶点,助力胰腺癌治疗药物的开发。

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L2192
产品编号: L2192
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品特点:
  • 2508种与胰腺癌相关的化合物,可以用于高通量和高内涵筛选;
  • 靶点含KRas, MEK, ERK, RAF, PI3K, HER2, EGFR, JAK/STAT, IGF-1R, VEGF, TGFβ等;
  • 部分化合物已上市或已进入临床期;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库组成
Apoptosis
Autophagy
NF-κB
PI3K
EGFR
CDK
COX
VEGFR
PPAR
Wnt/beta-catenin
mTOR
JAK
Akt
HDAC
PARP
STAT
Src
ERK
AMPK
GSK-3
FGFR
p38 MAPK
Endogenous Metabolite
Antibacterial
c-Met/HGFR
PDGFR
Raf
FLT
p53
TGF-beta/Smad
c-Kit
MEK
Potassium Channel
JNK
MMP
IGF-1R
Reactive Oxygen Species
TNF
Tyrosine Kinases
Caspase
Parasite
Ras
Bcr-Abl
DNA-PK
S6 Kinase
ATM/ATR
ALK
Aurora Kinase
Ferroptosis
HER
HIF/HIF Prolyl-Hydroxylase
MAPK
Cytochromes P450
DNA/RNA Synthesis
IL Receptor
Antibiotic
c-RET
Influenza Virus
Mdm2
PDK
Mitophagy
Pim
STING
Gamma-secretase
HIF
HIV Protease
Bcl-2 Family
E1/E2/E3 Enzyme
Hedgehog/Smoothened
PD-1/PD-L1
Kras
Antifungal
Lipoxygenase
PKC
Calcium Channel
PKA
Casein Kinase
Dehydrogenase
FAK
NO Synthase
Nrf2
PI4K
Prostaglandin Receptor
Topoisomerase
IκB/IKK
Trk receptor
Beta Amyloid
c-Fms
Chk
Epigenetic Reader Domain
NOS
PDE
Virus Protease
Rho
ROS
Interleukin
TAM Receptor
Tyrosinase
HSV
Phosphatase
Sirtuin
5-HT Receptor
Adrenergic Receptor
Antioxidant
HCV Protease
ROCK
SIK
Sodium Channel
Syk
Drug Metabolite
DYRK
GABA Receptor
Microtubule Associated
Mitochondrial Metabolism
Others
PGE Synthase
PTEN
AChR
Antifection
Anti-infection
Antiviral
Aryl Hydrocarbon Receptor
ATPase
CSF-1R
Ephrin Receptor
HSP
MLK
PERK
P-gp
PLK
Proteasome
Smo
TLR
Adenosine Receptor
Carbonic Anhydrase
Estrogen/progestogen Receptor
GPCR
IAP
Integrin
IRAK
MELK
RIP kinase
SGK
Tie-2
transporter
TRP/TRPV Channel
BTK
Cannabinoid Receptor
CCR
Chloride channel
Cholecystokinin Receptor
Cholinesterase (ChE)
c-Myc
Glucosidase
GTPase
HBV
Histamine Receptor
IFNAR
LDL
PYK2
ROS Kinase
Serine Protease
Serine/threonin kinase
Androgen Receptor
BACE
CaMK
cAMP
Decarboxylase
Discoidin Domain Receptor (DDR)
DNA Alkylation
DNA Alkylator/Crosslinker
DUB
Estrogen Receptor/ERR
Free radical scavengers
Glucocorticoid Receptor
Glutathione Peroxidase
Hck
Histone Methyltransferase
Leukotriene Receptor
LRRK2
MNK
MRP
NADPH
NMDAR
NOD
Opioid Receptor
Phospholipase
Porcupine
RAAS
Retinoid Receptor
SARS-CoV
Transferase
ABC Transporter
ACK1
Acyltransferase
ADC Cytotoxin
Aromatase
ATP Citrate Lyase
Beta-Secretase
Cell Cycle Arrest
Dopamine Receptor
FAAH
Gap Junction Protein
Glucokinase
GluR
Hippo pathway
Histone Acetyltransferase
Histone Demethylase
Immunology/Inflammation related
Lipid
NADPH-oxidase
NOD-like Receptor (NLR)
Nucleoside Antimetabolite/Analog
Progesterone Receptor
Proton pump
Reverse Transcriptase
RSV
S1P Receptor
UGT
Adenosine Deaminase
Adenylyl Cyclase
Aminopeptidase
Arginase
ASK
BCRP
BMI-1
CFTR
CRISPR/Cas9
Cysteine Protease
DAPK
DHFR
DNA
DNA Methyltransferase
DPP-4
Epoxide Hydrolase
Fatty Acid Synthase
FLAP
FXR
gp120/CD4
Guanylate cyclase
Haspin Kinase
hCE
Hexokinase
Hydroxylase
iGluR
IRE1
Kinesin
Liver X Receptor
LPA Receptor
LPL Receptor
LTR
Melanin-concentrating Hormone Receptor (MCHR)
Methionine Adenosyltransferase (MAT)
MicroRNA
Monoamine Transporter
Myosin
Na+/Ca2+ Exchanger
NPC1L1
OCT
p97
PAD
PAFR
PAI-1
PAK
PKM
Pyroptosis
RAR/RXR
Reductase
ROR
Sigma receptor
Thioredoxin
Thrombin
Thrombopoietin Receptor
TOPK
VDA
YAP
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