自噬库

Autophagy Compound Library
产品编号: L3200

自噬是一个涉及到细胞自身物质或结构被溶酶体或液泡分解的过程。先是内质网脱落的双层膜包裹细胞内部分受损或老化的细胞器、蛋白质等成分形成自噬体,后与溶酶体或液泡融合降解其所包裹的内容物,以实现细胞本身的代谢需要和某些细胞器的更新。细胞自噬与细胞凋亡、细胞衰老一样,是十分重要的生物学现象,参与生物的发育、生长等多种过程,细胞自噬的异常导致癌细胞的出现。 TargetMol 自噬库集合了文献报道的 1470 种细胞自噬相关的生物活性小分子化合物,可用于细胞自噬机理研究和靶向药物筛选。

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L3200
产品编号: L3200
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
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技术资料
产品描述
产品描述:
  • 1470种细胞自噬相关的生物活性小分子化合物的特有集合,用于自噬相关的研究,用于高通量、高内涵筛选 ;
  • 产品经过临床验证和临床实验,具有生物安全保障和一定的生物活性 ;
  • 是研究细胞自噬的机理以及药物靶向研究的有效工具 ;
  • 活性包括自噬诱导、自噬抑制、蛋白酶体、HIF、E3 Ligase、mTOR等 ;
  • 结构多样,药效显著,可渗透细胞 ;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等 ;
  • NMR和HPLC检测技术保证产品高纯度和高质量 ;
  • 所有化合物现货供应。
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化合物库组成
Autophagy
Apoptosis
PI3K
mTOR
Akt
Antibacterial
AMPK
GSK-3
Endogenous Metabolite
Antibiotic
CDK
Mitophagy
p38 MAPK
CXCR
NF-κB
HDAC
HIV Protease
DNA-PK
ERK
Parasite
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Reactive Oxygen Species
Raf
S6 Kinase
VEGFR
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ATM/ATR
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DNA/RNA Synthesis
PDK
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COX
Cytochromes P450
PKC
Src
Bcr-Abl
LRRK2
Retinoid Receptor
EGFR
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Calcium Channel
c-Kit
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Aurora Kinase
Caspase
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PPAR
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Dehydrogenase
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FXR
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JAK
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Nrf2
PDE
HSV
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PERK
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IGF-1R
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p53
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TGF-beta/Smad
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SIK
Sirtuin
Sodium Channel
TRP/TRPV Channel
ALK
Antioxidant
ATPase
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GABA Receptor
HIF
HSP
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PTEN
Rho
Beta Amyloid
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transporter
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ribosome
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GPCR
HER
Histone Acetyltransferase
IAP
iGluR
IRE1
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Mdm2
MLK
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Monoamine Transporter
NMDAR
NOD-like Receptor (NLR)
Norepinephrine
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RAR/RXR
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ACK1
Acyltransferase
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Aminopeptidase
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BCRP
cAMP
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IDO
Imidazoline Receptor
Immunology/Inflammation related
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IRAK
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