普林斯顿生物分子研究中的 Fsp3富集库包含11089个化合物。片段(Fragments)仍然非常受欢迎,并将至少保持3-5年的需求。创建几个片段库相当简单和快速,例如:通用片段(分子量≤300,ClogP≤3,HbD≤3,去除不需要的功能基团),氟化片段(用于核磁共振筛选),黄金集(Ro3和 Veber 规则,应用了 PAINS 和 Lilly MedChem 规则)。普林斯顿生物分子研究中的 Fsp3富集库包含11089个化合物。
Fragments are still in high demand and would stay for at least 3-5 years. It is quite easy and fast to create few fragments libraries, e.g.: General Fragments (MW ≤ 300, ClogP ≤ 3, HbD ≤ 3, undesired functionalities removed), Fluorinated Fragments (for NMR screening), Golden set (Ro3 & Veber rules, PAINS + Lilly MedChem rules applied). Fsp3 enriched Library in the Princeton BioMolecal Research contains 11089 compounds.