神经保护化合物库

Neuroprotective Compound Library
产品编号: L2640

神经保护(Neuroprotection)是指通过各种机制和手段来防止神经元受到损伤或促进神经元的修复,从而保护神经系统功能的过程。这一领域的研究主要集中在防止神经元凋亡、减少炎症反应、减少氧化应激和促进神经再生等方面。神经保护在许多神经退行性疾病(如阿尔茨海默病、帕金森病、多发性硬化症)以及急性神经损伤(如中风和脊髓损伤)中具有重要意义。研究揭示了多个关键靶点,如抗氧化,神经营养因子,钙离子通道等在预防神经元损伤、促进神经再生以及对抗神经退行性疾病方面展现出潜力。 TargetMol神经保护化合物库收集了1120种具有神经保护活性及潜在的神经保护活性化合物,可用于神经保护相关的药物研发,神经保护相关机制探索。

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L2640
产品编号: L2640
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
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技术资料
产品描述
产品描述:
  • 1120种神经保护相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
  • 靶点包括BDNF、Calcium Channel、Sodium Channel、NMDAR/TRPM4等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
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化合物库组成
Calcium Channel
Sodium Channel
Wnt/beta-catenin
Apoptosis
Potassium Channel
GSK-3
Others
NO Synthase
GABA Receptor
Autophagy
Endogenous Metabolite
iGluR
NMDAR
GluR
AMPK
NF-κB
Antibacterial
Reactive Oxygen Species
COX
AChR
CDK
NOS
Antioxidant
Cytochromes P450
Akt
5-HT Receptor
TNF
PARP
Parasite
Beta Amyloid
Dopamine Receptor
ERK
IL Receptor
Caspase
TRP/TRPV Channel
PDE
ROS
Cholinesterase (ChE)
PI3K
Mitophagy
PPAR
p38 MAPK
Adenosine Receptor
Histamine Receptor
Adrenergic Receptor
MAO
Prostaglandin Receptor
PKC
Influenza Virus
EGFR
Bcl-2 Family
Tyrosinase
Antibiotic
HIF/HIF Prolyl-Hydroxylase
RAAS
JNK
PKA
mTOR
Interleukin
STAT
S6 Kinase
HER
Monoamine Oxidase
ATPase
HIV Protease
Carbonic Anhydrase
Src
Phosphatase
Virus Protease
Mitochondrial Metabolism
JAK
HSV
MMP
MAPK
P-gp
Nrf2
GPR
MEK
Anti-infection
Microtubule Associated
Ferroptosis
Na+/Ca2+ Exchanger
Serine/threonin kinase
Glucocorticoid Receptor
Gamma-secretase
Glucosidase
Antifection
Aurora Kinase
Epigenetic Reader Domain
Lipoxygenase
TGF-beta/Smad
Lipid
DNA/RNA Synthesis
Porcupine
Casein Kinase
NOD
Sigma receptor
Estrogen/progestogen Receptor
Antifungal
Estrogen Receptor/ERR
Serotonin Transporter
VEGFR
E1/E2/E3 Enzyme
LDL
Drug Metabolite
Opioid Receptor
Chk
Norepinephrine
CaMK
Beta-Secretase
Antiviral
TLR
Trk receptor
transporter
HDAC
Cannabinoid Receptor
FLT
HMG-CoA Reductase
Imidazoline Receptor
S1P Receptor
Chloride channel
HCV Protease
Integrin
Arginase
LPL Receptor
BACE
Reductase
DYRK
PERK
Cysteine Protease
ROCK
Immunology/Inflammation related
Topoisomerase
Bcr-Abl
P2X Receptor
Monoamine Transporter
Guanylate cyclase
PTEN
Somatostatin
Xanthine Oxidase
cAMP
IGF-1R
PGE Synthase
SARS-CoV
LRRK2
Sirtuin
Pyroptosis
IκB/IKK
PDK
Phospholipase
HIF
FGFR
Ras
AhR
p53
Thyroid hormone receptor(THR)
Proteasome
Adenylyl Cyclase
DHFR
Piezo Channel
Amino Acids and Derivatives
Dehydrogenase
YAP
Arrestin
gp120/CD4
GTPase
Progesterone Receptor
OCT
MRP
HBV
Cholecystokinin Receptor
Tyrosine Kinases
Cell Cycle Arrest
NAMPT
Glucokinase
Amylase
Aryl Hydrocarbon Receptor
CSF-1R
Myosin
UGT
PAFR
Raf
DNA gyrase
HCN Channel
DPP-4
Fatty Acid Synthase
PDGFR
Stearoyl-CoA Desaturase (SCD)
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Telomerase
ATP Citrate Lyase
RSV
Methionine Adenosyltransferase (MAT)
GST
Acetyl-CoA Carboxylase
Retinoid Receptor
ribosome
Adenosine Deaminase
DNA Methyltransferase
NADPH-oxidase
TAM Receptor
ROS Kinase
Sodium-dependent phosphate transporter
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