神经递质受体化合物库

Neurotransmitter Receptor Compound Library
产品编号: L2610

神经递质是人类行为的化学基础。研究证实行为病理大都由一个或数个神经递质缺失或增多失平衡引起。躯体疾病也可由于特殊的神经径路障碍引起,例如帕金森病(PD)。脑内神经递质分为生物原胺类、氨基酸类、肽类、乙酰胆碱类等。生物原胺类神经递质包括:多巴胺(DA)、去甲肾上腺素(NE)、肾上腺素(E)、5-羟色胺(5-HT)也称(血清素)。氨基酸类神经递质包括:γ-氨基丁酸(GABA)、甘氨酸、谷氨酸、组胺。肽类神经递质分为:内源性阿片肽、P 物质、神经加压素、胆囊收缩素(CCK)、生长抑素、血管加压素和缩宫素、神经肽 Y。其它神经递质还有:核苷酸类、花生酸碱、阿南德酰胺、sigma 受体(σ受体)。在突触后膜或效应器细胞膜上有能与神经递质相结合的特殊蛋白质,称神经递质受体或突触后受体。许多精神药物作用于神经递质受体。 TargetMol 收集了 1660 种神经递质受体相关的化合物,可用于神经系统药物的开发。

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L2610
产品编号: L2610
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
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技术资料
产品描述
产品描述:
  • 1660种与神经递质受体相关的化合物,用于高通量、高内涵筛选;
  • 靶点包括5-HT receptor、AChR、GABA receptor、dopamine receptor、Opiod receptor等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、活性描述等;
  • NMR、HPLC/LCMS等多种检测技术保证产品结构正确,纯度高,减少假阳性。
化合物库定制
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化合物库组成
5-HT Receptor
AChR
Adrenergic Receptor
Dopamine Receptor
Histamine Receptor
GABA Receptor
Adenosine Receptor
GluR
NMDAR
iGluR
Autophagy
Endogenous Metabolite
Norepinephrine
Apoptosis
Serotonin Transporter
Calcium Channel
Potassium Channel
Sodium Channel
Antibacterial
Cholinesterase (ChE)
PDE
Cytochromes P450
Parasite
Influenza Virus
Sigma receptor
TRP/TRPV Channel
CaMK
HIV Protease
Antibiotic
HCV Protease
HER
NF-κB
Reactive Oxygen Species
Antifungal
HDAC
MAO
ABC Transporter
BACE
COX
Dehydrogenase
DNA/RNA Synthesis
Drug Metabolite
ERK
Ferroptosis
Histone Methyltransferase
Lipoxygenase
Mitophagy
Monoamine Transporter
NO Synthase
Opioid Receptor
P2X Receptor
P-gp
Phospholipase
TNF
AMPK
Beta Amyloid
cAMP
Cannabinoid Receptor
Caspase
Chloride channel
Glucocorticoid Receptor
GPR
Imidazoline Receptor
Monoamine Oxidase
MRP
PI3K
PKA
Prostaglandin Receptor
RAAS
ROS
SARS-CoV
Transferase
VEGFR
Virus Protease
Acyltransferase
Adenylyl Cyclase
Antifection
Anti-infection
Antioxidant
Aurora Kinase
Bcl-2 Family
Beta-Secretase
EGFR
Gamma-secretase
GSK-3
IL Receptor
Immunology/Inflammation related
MEK
Melatonin Receptor
MT Receptor
NOS
PAFR
PARP
Phosphatase
Platelet aggregation
PPAR
STAT
Transaminase
Tyrosinase
ACK1
Adenosine Deaminase
Adiponectin Receptor
Akt
Amino Acids and Derivatives
Aminopeptidase
Androgen Receptor
Angiotensin-converting Enzyme (ACE)
Annexin A
Antifolate
Arrestin
Aryl Hydrocarbon Receptor
ATM/ATR
Bcr-Abl
Bombesin Receptor
Carbonic Anhydrase
CCR
CDK
CRISPR/Cas9
DNA
DNA Methyltransferase
DYRK
Epigenetic Reader Domain
FAK
Fatty Acid Synthase
FGFR
FLT
FXR
Gap Junction Protein
GluCls
Glucosidase
GlyT
GRK
GST
GTPase
HBV
HCN Channel
HIF/HIF Prolyl-Hydroxylase
HMG-CoA Reductase
HSV
Hydroxylase
IAP
Indoleamine 2,3-Dioxygenase (IDO)
Integrin
Interleukin
LDL
Leukotriene Receptor
LTR
Melanin-concentrating Hormone Receptor (MCHR)
Microtubule Associated
Mitochondrial Metabolism
MMP
mTOR
Na+/Ca2+ Exchanger
NADPH
NOD
OCT
Others
p38 MAPK
p53
PAD
PKC
Raf
Reductase
Reverse Transcriptase
RSV
Stearoyl-CoA Desaturase (SCD)
Syk
TGF-beta/Smad
transporter
Trk receptor
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