核受体化合物库

Nuclear Receptor Compound Library
产品编号: L1510

核受体是细胞内一类区别于膜受体的蛋白,它们与相应配体结合后,能够直接与基因组DNA 结合并调节相邻基因表达,因此这类受体被归类为转录因子。核受体在胚胎发育和机体内环境平衡中发挥关键作用。近年来,核受体家族在代谢性疾病领域受到广泛的关注,已有研究证明,它们与糖尿病、脂肪肝等疾病的发生发展密切相关,也被称为代谢性核受体。 TargetMol 汇集了631 种有文献报道的核受体相关化合物,适用于核受体相关信号通路及疾病研究,可用于高通量筛选和高内涵筛选。

陶术生物的所有产品和服务仅用于科学研究,我们不为任何个人用途提供产品和服务。
L1510
产品编号: L1510
规格
1 mg
30 μL x 10 mM (in DMSO)
50 μL x 10 mM (in DMSO)
100 μL x 10 mM (in DMSO)
250 μL x 10 mM (in DMSO)
特别折扣
等您来询问!
技术资料
产品描述
产品描述:
  • 631个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选;
  • 提供产品的来源、化学信息和生物学信息,为筛选提供理论方向和研究基础;
  • 结构多样,药效显著,可渗透细胞;
  • NMR和HPLC技术保证产品高纯度。
化合物库定制
我们的化合物库可以灵活定制! 了解更多
化合物库咨询
验证码
化合物库组成
PPAR
Estrogen/progestogen Receptor
Estrogen Receptor/ERR
Androgen Receptor
Autophagy
Glucocorticoid Receptor
Endogenous Metabolite
Retinoid Receptor
Apoptosis
Progesterone Receptor
Others
FXR
ROR
Thyroid hormone receptor(THR)
AhR
COX
Liver X Receptor
Antibacterial
NF-κB
Cytochromes P450
Aryl Hydrocarbon Receptor
Reactive Oxygen Species
TSH Receptor
Antifungal
Ferroptosis
GPR
Akt
AMPK
Antibiotic
IL Receptor
Potassium Channel
RAR/RXR
Adrenergic Receptor
Bcl-2 Family
Drug Metabolite
GPCR19
Influenza Virus
Lipoxygenase
MMP
Parasite
Prostaglandin Receptor
Reductase
TNF
Tyrosinase
Annexin A
Calcium Channel
Cannabinoid Receptor
Epigenetic Reader Domain
Interleukin
Mitochondrial Metabolism
Mitophagy
NO Synthase
Nrf2
p38 MAPK
p53
ROS
SARS-CoV
ADC Cytotoxin
ABC Transporter
AChR
Antioxidant
Aromatase
ERK
GABA Receptor
Glutathione Peroxidase
GSK-3
HIV Protease
JNK
NOS
PARP
PDE
Phosphatase
Sirtuin
Smo
transporter
TRP/TRPV Channel
VEGFR
Virus Protease
Wnt/beta-catenin
Adenylyl Cyclase
Antifection
CaMK
Carbonic Anhydrase
Caspase
c-Kit
c-Met/HGFR
Complement System
Cysteine Protease
Dehydrogenase
DNA
DNA Methyltransferase
DNA/RNA Synthesis
EGFR
Epoxide Hydrolase
Fatty Acid Synthase
FLAP
FLT
Gamma-secretase
Glucagon Receptor
Glucokinase
Glucosidase
GluR
GNRH Receptor
gp120/CD4
HBV
HCV Protease
HER
HIF/HIF Prolyl-Hydroxylase
Histamine Receptor
Histone Acetyltransferase
Histone Methyltransferase
HMG-CoA Reductase
HSP
Hydroxylase
IFNAR
Immunology/Inflammation related
LDL
Leukotriene Receptor
Lipid
MAO
Melatonin Receptor
MRP
mTOR
Nucleoside Antimetabolite/Analog
Opioid Receptor
PAK
PERK
P-gp
Phospholipase
Phosphorylase
PKA
PKC
Proteasome
RAAS
S1P Receptor
Sodium Channel
STAT
STING
TAM Receptor
Thrombin
Topoisomerase
PGC-1α
化合物库信息示例
Empty981-15-797322-87-7959-23-995853-92-2958323-31-4958295-17-5956104-40-895167-41-2950-99-294987-08-3Empty
AilanthoneTroglitazone4'-MethoxychalconeCGS 15435TLX agonist 1AGN 196996ApalutamideDY1312,2,5,7,8-Pentamethyl-6-ChromanolGypenoside XLIX
Empty945966-46-1945619-74-994497-51-594105-90-593987-29-2936345-35-6936345-34-5931314-31-7929492-71-7928134-65-0Empty
ApararenoneOPHIOPOGONIN DTamibarotene(±)-EquolBI-6015PF-02413873Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl-Specific PXR antagonist 70GAC0003A4Osilodrostat
Empty927961-18-0926228-58-2923978-27-2920509-32-6915087-33-1915087-27-3912789-08-3905954-18-9904449-84-990357-06-5Empty
LanifibranorCTK8A3536ElafibranorResmetiromEnzalutamideRD162ISX-3IsopsoralenosideNR2F6 modulator-1Bicalutamide
Empty899821-23-9898800-26-589778-26-789-57-6895542-09-388678-67-5882-09-7881639-98-1880635-03-0877387-37-6Empty
ACP-105AZ876Toremifene5-Aminosalicylic AcidtrifarotenePyributicarbClofibric acidG-1GW6471GSK5182
Empty875787-07-8870888-46-3870773-76-5870554-67-9863588-32-3863239-61-6863239-60-5862907-48-086111-26-4856676-23-8Empty
LXR-623AC-262536AC-261066GQ-16ML-180Tauro-Obeticholic acidGlyco-Obeticholic acidAH-3960ZindoxifeneCholine Fenofibrate
Empty85666-24-685666-17-7853-23-6852948-13-1851983-85-2851528-79-5851107-28-3850-52-2849662-80-2848259-27-8Empty
FuregrelateFuregrelate sodiumDehydroisoandrosterone 3-acetateMB-07811GaleteroneSeladelparCMP8AltrenogestY134Pemafibrate
Empty848142-62-1847239-17-284687-43-484371-65-384-17-384-16-2841205-47-8839673-52-883919-23-7835619-41-5Empty
Indazole-ClUVI 3003Astragaloside IVMifepristoneDienestrolHexestrolOstarineCevoglitazarMometasone furoateIndeglitazar
Empty83-49-883-34-1827319-43-782640-04-8824932-88-982413-20-582034-46-681485-25-880-92-2805239-56-9Empty
Hyodeoxycholic acidSkatoleGW-870086Raloxifene hydrochloride(E/Z)-ElafibranorDroloxifeneLoteprednol etabonatePeretinoinPregnanediolPHTPP
TargetMol | Target Loading
正在加载 ~