核受体是细胞内一类区别于膜受体的蛋白,它们与相应配体结合后,能够直接与基因组DNA 结合并调节相邻基因表达,因此这类受体被归类为转录因子。核受体在胚胎发育和机体内环境平衡中发挥关键作用。近年来,核受体家族在代谢性疾病领域受到广泛的关注,已有研究证明,它们与糖尿病、脂肪肝等疾病的发生发展密切相关,也被称为代谢性核受体。 TargetMol 汇集了631 种有文献报道的核受体相关化合物,适用于核受体相关信号通路及疾病研究,可用于高通量筛选和高内涵筛选。
Empty | 981-15-7 | 97322-87-7 | 959-23-9 | 95853-92-2 | 958323-31-4 | 958295-17-5 | 956104-40-8 | 95167-41-2 | 950-99-2 | 94987-08-3 | Empty |
Ailanthone | Troglitazone | 4'-Methoxychalcone | CGS 15435 | TLX agonist 1 | AGN 196996 | Apalutamide | DY131 | 2,2,5,7,8-Pentamethyl-6-Chromanol | Gypenoside XLIX | ||
Empty | 945966-46-1 | 945619-74-9 | 94497-51-5 | 94105-90-5 | 93987-29-2 | 936345-35-6 | 936345-34-5 | 931314-31-7 | 929492-71-7 | 928134-65-0 | Empty |
Apararenone | OPHIOPOGONIN D | Tamibarotene | (±)-Equol | BI-6015 | PF-02413873 | Benzonitrile, 4-[[5-cyclopropyl-3-methyl-1-[(methylsulfonyl)methyl]-1H-pyrazol-4-yl]oxy]-2,6-dimethyl- | Specific PXR antagonist 70 | GAC0003A4 | Osilodrostat | ||
Empty | 927961-18-0 | 926228-58-2 | 923978-27-2 | 920509-32-6 | 915087-33-1 | 915087-27-3 | 912789-08-3 | 905954-18-9 | 904449-84-9 | 90357-06-5 | Empty |
Lanifibranor | CTK8A3536 | Elafibranor | Resmetirom | Enzalutamide | RD162 | ISX-3 | Isopsoralenoside | NR2F6 modulator-1 | Bicalutamide | ||
Empty | 899821-23-9 | 898800-26-5 | 89778-26-7 | 89-57-6 | 895542-09-3 | 88678-67-5 | 882-09-7 | 881639-98-1 | 880635-03-0 | 877387-37-6 | Empty |
ACP-105 | AZ876 | Toremifene | 5-Aminosalicylic Acid | trifarotene | Pyributicarb | Clofibric acid | G-1 | GW6471 | GSK5182 | ||
Empty | 875787-07-8 | 870888-46-3 | 870773-76-5 | 870554-67-9 | 863588-32-3 | 863239-61-6 | 863239-60-5 | 862907-48-0 | 86111-26-4 | 856676-23-8 | Empty |
LXR-623 | AC-262536 | AC-261066 | GQ-16 | ML-180 | Tauro-Obeticholic acid | Glyco-Obeticholic acid | AH-3960 | Zindoxifene | Choline Fenofibrate | ||
Empty | 85666-24-6 | 85666-17-7 | 853-23-6 | 852948-13-1 | 851983-85-2 | 851528-79-5 | 851107-28-3 | 850-52-2 | 849662-80-2 | 848259-27-8 | Empty |
Furegrelate | Furegrelate sodium | Dehydroisoandrosterone 3-acetate | MB-07811 | Galeterone | Seladelpar | CMP8 | Altrenogest | Y134 | Pemafibrate | ||
Empty | 848142-62-1 | 847239-17-2 | 84687-43-4 | 84371-65-3 | 84-17-3 | 84-16-2 | 841205-47-8 | 839673-52-8 | 83919-23-7 | 835619-41-5 | Empty |
Indazole-Cl | UVI 3003 | Astragaloside IV | Mifepristone | Dienestrol | Hexestrol | Ostarine | Cevoglitazar | Mometasone furoate | Indeglitazar | ||
Empty | 83-49-8 | 83-34-1 | 827319-43-7 | 82640-04-8 | 824932-88-9 | 82413-20-5 | 82034-46-6 | 81485-25-8 | 80-92-2 | 805239-56-9 | Empty |
Hyodeoxycholic acid | Skatole | GW-870086 | Raloxifene hydrochloride | (E/Z)-Elafibranor | Droloxifene | Loteprednol etabonate | Peretinoin | Pregnanediol | PHTPP |